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Safety and Pharmacokinetics of Single-Dose Novel Oral Androgen 11β-Methyl-19-Nortestosterone-17β-Dodecylcarbonate in Men

CONTEXT: 11β-Methyl-19-nortestosterone-17β-dodecylcarbonate (11β-MNTDC) is an orally bioavailable prodrug of 11β-methyl-19-nortestosterone (11β-MNT) with androgenic and progestational activity. OBJECTIVES: (i) Quantify 11β-MNT binding to androgen and progesterone receptors. (ii) Evaluate safety, tol...

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Bibliografski detalji
Izdano u:J Clin Endocrinol Metab
Glavni autori: Wu, Sherry, Yuen, Fiona, Swerdloff, Ronald S, Pak, Youngju, Thirumalai, Arthi, Liu, Peter Y, Amory, John K, Bai, Feng, Hull, Laura, Blithe, Diana L, Anawalt, Bradley D, Parman, Toufan, Kim, Kyuri, Lee, Min S, Bremner, William J, Page, Stephanie T, Wang, Christina
Format: Artigo
Jezik:Inglês
Izdano: Endocrine Society 2018
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC6334268/
https://ncbi.nlm.nih.gov/pubmed/30252057
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1210/jc.2018-01528
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