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Enhanced Tumor Selectivity of 5-Fluorouracil Using a Reactive Oxygen Species-Activated Prodrug Approach

[Image: see text] We report the design, synthesis, and evaluation of novel 5-fluorouracil (5FU) prodrugs 1a,1b that are efficiently activated by the high level of reactive oxygen species (ROS) in cancer cells. Prodrugs 1a,1b selectively kill cancer cells over normal cells and are well-tolerated in m...

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Detalles Bibliográficos
Publicado en:ACS Med Chem Lett
Autores principales: Ai, Yong, Obianom, Obinna N., Kuser, Meredith, Li, Yue, Shu, Yan, Xue, Fengtian
Formato: Artigo
Lenguaje:Inglês
Publicado: American Chemical Society 2018
Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC6331168/
https://ncbi.nlm.nih.gov/pubmed/30655959
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsmedchemlett.8b00539
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