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Activation of 2,4-Diaminoquinazoline in Mycobacterium tuberculosis by Rv3161c, a Putative Dioxygenase

The diaminoquinazoline series has good potency against Mycobacterium tuberculosis. Resistant isolates have mutations in Rv3161c, a putative dioxygenase. We carried out metabolite analysis on a wild-type strain and an Rv3161c mutant strain after exposure to a diaminoquinazoline. The parental compound...

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Bibliografski detalji
Izdano u:Antimicrob Agents Chemother
Glavni autori: Melief, Eduard, Bonnett, Shilah A., Zuniga, Edison S., Parish, Tanya
Format: Artigo
Jezik:Inglês
Izdano: American Society for Microbiology 2018
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC6325208/
https://ncbi.nlm.nih.gov/pubmed/30323042
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.01505-18
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