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Brain Distribution and Metabolism of Flupirtine, a Nonopioid Analgesic Drug with Antiseizure Effects, in Neonatal Rats

Flupirtine, a nonopioid analgesic drug, is effective in treating neonatal seizures. However, its brain delivery and pharmacokinetics are unknown in neonatal mammals. The purpose of this study was to determine the pharmacokinetics of flupirtine and the formation of its active metabolite D-13223 in va...

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Dettagli Bibliografici
Pubblicato in:Pharmaceutics
Autori principali: Patil, Madhoosudan A., Matter, Brock A., Raol, Yogendra H., Bourne, David W. A., Kelley, Ryan A., Kompella, Uday B.
Natura: Artigo
Lingua:Inglês
Pubblicazione: MDPI 2018
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6320943/
https://ncbi.nlm.nih.gov/pubmed/30558371
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/pharmaceutics10040281
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