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Analgesic Activity of Acid-Sensing Ion Channel 3 (ASIС3) Inhibitors: Sea Anemones Peptides Ugr9-1 and APETx2 versus Low Molecular Weight Compounds

Acid-sensing ion channel 3 (ASIC3) makes an important contribution to the development and maintenance of inflammatory and acid-induced pain. We compared different ASIC3 inhibitors (peptides from sea anemones (APETx2 and Ugr9-1) and nonpeptide molecules (sevanol and diclofenac)) in anti-inflammatory...

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Detalhes bibliográficos
Publicado no:Mar Drugs
Main Authors: Andreev, Yaroslav A., Osmakov, Dmitry I., Koshelev, Sergey G., Maleeva, Ekaterina E., Logashina, Yulia A., Palikov, Victor A., Palikova, Yulia A., Dyachenko, Igor A., Kozlov, Sergey A.
Formato: Artigo
Idioma:Inglês
Publicado em: MDPI 2018
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6316600/
https://ncbi.nlm.nih.gov/pubmed/30545037
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/md16120500
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