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Generation of inhibitory monoclonal antibodies targeting matrix metalloproteinase-14 by motif grafting and CDR optimization

Matrix metalloproteinase-14 (MMP-14) plays important roles in cancer metastasis, and the failures of broad-spectrum MMP compound inhibitors in clinical trials suggested selectivity is critical. By grafting an MMP-14 specific inhibition motif into complementarity determining region (CDR)-H3 of antibo...

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Publicat a:Protein Eng Des Sel
Autors principals: Nam, Dong Hyun, Fang, Kuili, Rodriguez, Carlos, Lopez, Tyler, Ge, Xin
Format: Artigo
Idioma:Inglês
Publicat: Oxford University Press 2017
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6283398/
https://ncbi.nlm.nih.gov/pubmed/27986919
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1093/protein/gzw070
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