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Design, Synthesis and Biological Evaluation of Novel Benzothiazole Derivatives as Selective PI3Kβ Inhibitors

A novel series of PI3Kβ (Phosphatidylinositol-3-kinases beta subunit) inhibitors with the structure of benzothiazole scaffold have been designed and synthesized. All the compounds have been evaluated for inhibitory activities against PI3Kα, β, γ, δ and mTOR (Mammalian target of rapamycin). Two super...

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Detalles Bibliográficos
Publicado en:Molecules
Main Authors: Cao, Shuang, Cao, Ruiyuan, Liu, Xialing, Luo, Xiang, Zhong, Wu
Formato: Artigo
Idioma:Inglês
Publicado: MDPI 2016
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC6274018/
https://ncbi.nlm.nih.gov/pubmed/27384552
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules21070876
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