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Osimertinib (AZD9291), a Mutant-Selective EGFR Inhibitor, Reverses ABCB1-Mediated Drug Resistance in Cancer Cells

In recent years, tyrosine kinase inhibitors (TKIs) have been shown capable of inhibiting the ATP-binding cassette (ABC) transporter-mediated multidrug resistance (MDR). In this study, we determine whether osimertinib, a novel selective, irreversible EGFR (epidermal growth factor receptor) TKI, could...

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Gorde:
Xehetasun bibliografikoak
Argitaratua izan da:Molecules
Egile Nagusiak: Zhang, Xiao-Yu, Zhang, Yun-Kai, Wang, Yi-Jun, Gupta, Pranav, Zeng, Leli, Xu, Megan, Wang, Xiu-Qi, Yang, Dong-Hua, Chen, Zhe-Sheng
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: MDPI 2016
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC6273565/
https://ncbi.nlm.nih.gov/pubmed/27649127
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules21091236
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