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Antibacterial Barbituric Acid Analogues Inspired from Natural 3-Acyltetramic Acids; Synthesis, Tautomerism and Structure and Physicochemical Property-Antibacterial Activity Relationships

The synthesis, tautomerism and antibacterial activity of novel barbiturates is reported. In particular, 3-acyl and 3-carboxamidobarbiturates exhibited antibacterial activity, against susceptible and some resistant Gram-positive strains of particular interest is that these systems possess amenable mo...

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Publicado en:Molecules
Main Authors: Jeong, Yong-Chul, Moloney, Mark G.
Formato: Artigo
Idioma:Inglês
Publicado: MDPI 2015
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC6272196/
https://ncbi.nlm.nih.gov/pubmed/25710842
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules20033582
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