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Receptor-Based Virtual Screening of EGFR Kinase Inhibitors from the NCI Diversity Database

Epidermal growth factor receptor (EGFR) abnormalities have been associated with several types of human cancer. The crystal structures of its tyrosine kinase domain (EGFR-TK) complexed with small molecule inhibitors revealed the kinase inhibition modes, prompting us to search for novel anti-cancer dr...

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Dettagli Bibliografici
Pubblicato in:Molecules
Autori principali: Choowongkomon, Kiattawee, Sawatdichaikul, Orathai, Songtawee, Napat, Limtrakul, Jumras
Natura: Artigo
Lingua:Inglês
Pubblicazione: MDPI 2010
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6264413/
https://ncbi.nlm.nih.gov/pubmed/20657425
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules15064041
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