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B-973, a Novel α7 nAChR Ago-PAM: Racemic and Asymmetric Synthesis, Electrophysiological Studies, and in Vivo Evaluation

[Image: see text] We report here the total synthesis of B-973 (five steps), a recently identified α7 nAChR ago-PAM, its enantiomeric resolution, and its electrophysiological characterization in Xenopus oocytes to identify (−)-B-973B as the bioactive enantiomer. The asymmetric synthesis of B-973B was...

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Detalhes bibliográficos
Publicado no:ACS Med Chem Lett
Main Authors: Garai, Sumanta, Raja, Krishnamohan S., Papke, Roger L., Deschamps, Jeffrey R., Damaj, M. Imad, Thakur, Ganesh A.
Formato: Artigo
Idioma:Inglês
Publicado em: American Chemical Society 2018
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6231182/
https://ncbi.nlm.nih.gov/pubmed/30429960
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsmedchemlett.8b00407
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