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In Vivo Brain Imaging, Biodistribution, and Radiation Dosimetry Estimation of [(11)C]Celecoxib, a COX-2 PET Ligand, in Nonhuman Primates

COX-2 selective inhibitors (COXIBs) are non-steroidal anti-inflammatory drugs (NSAIDs), with fewer side effects compared with non-selective NSAIDs, and are used for the treatment of arthritis, headaches, and other inflammatory diseases of the brain and peripheral tissues. Radiolabeled COXIBs may per...

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Dades bibliogràfiques
Publicat a:Molecules
Autors principals: Kumar, J. S. Dileep, Bai, Bing, Zanderigo, Francesca, DeLorenzo, Christine, Prabhakaran, Jaya, Parsey, Ramin V., Mann, J. John
Format: Artigo
Idioma:Inglês
Publicat: MDPI 2018
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6222548/
https://ncbi.nlm.nih.gov/pubmed/30072617
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules23081929
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