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Heat shock protein 90 inhibitors overcome the resistance to Fms-like tyrosine kinase 3 inhibitors in acute myeloid leukemia

Internal tandem duplication (ITD) in Fms-like tyrosine kinase 3 (FLT3) is frequently observed in acute myeloid leukemia (AML). Quizartinib, gilteritinib, and midostaurin are inhibitors against FLT3-ITD that have good efficacy for FLT3-ITD-positive AML patients. Long-term administration leads to drug...

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Detalhes bibliográficos
Publicado no:Oncotarget
Main Authors: Katayama, Kazuhiro, Noguchi, Kohji, Sugimoto, Yoshikazu
Formato: Artigo
Idioma:Inglês
Publicado em: Impact Journals LLC 2018
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6188142/
https://ncbi.nlm.nih.gov/pubmed/30344940
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.18632/oncotarget.26045
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