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Making Sense of Pharmacology: Inverse Agonism and Functional Selectivity
Constitutive receptor activity/inverse agonism and functional selectivity/biased agonism are 2 concepts in contemporary pharmacology that have major implications for the use of drugs in medicine and research as well as for the processes of new drug development. Traditional receptor theory postulated...
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| Pubblicato in: | Int J Neuropsychopharmacol |
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| Autori principali: | , |
| Natura: | Artigo |
| Lingua: | Inglês |
| Pubblicazione: |
Oxford University Press
2018
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| Soggetti: | |
| Accesso online: | https://ncbi.nlm.nih.gov/pmc/articles/PMC6165953/ https://ncbi.nlm.nih.gov/pubmed/30085126 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1093/ijnp/pyy071 |
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