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Naphthalimides Selectively Inhibit the Activity of Bacterial, Replicative DNA Ligases and Display Bactericidal Effects against Tubercle Bacilli

The DNA ligases, enzymes that seal breaks in the backbones of DNA, are essential for all organisms, however bacterial ligases essential for DNA replication use β-nicotinamide adenine dinucleotide as their co-factor, whereas those that are essential in eukaryotes and viruses use adenosine-5′-triphosp...

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Detalhes bibliográficos
Publicado no:Molecules
Main Authors: Korycka-Machala, Malgorzata, Nowosielski, Marcin, Kuron, Aneta, Rykowski, Sebastian, Olejniczak, Agnieszka, Hoffmann, Marcin, Dziadek, Jaroslaw
Formato: Artigo
Idioma:Inglês
Publicado em: MDPI 2017
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6155577/
https://ncbi.nlm.nih.gov/pubmed/28106753
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules22010154
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