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Structure-Based Drug Design and Characterization of Sulfonyl-Piperazine Benzothiazinone Inhibitors of DprE1 from Mycobacterium tuberculosis

Macozinone (MCZ) is a tuberculosis (TB) drug candidate that specifically targets the essential flavoenzyme DprE1, thereby blocking synthesis of the cell wall precursor decaprenyl phosphoarabinose (DPA) and provoking lysis of Mycobacterium tuberculosis. As part of the MCZ backup program, we exploited...

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Detalhes bibliográficos
Publicado no:Antimicrob Agents Chemother
Main Authors: Piton, Jérémie, Vocat, Anthony, Lupien, Andréanne, Foo, Caroline S., Riabova, Olga, Makarov, Vadim, Cole, Stewart T.
Formato: Artigo
Idioma:Inglês
Publicado em: American Society for Microbiology 2018
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6153800/
https://ncbi.nlm.nih.gov/pubmed/30012754
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.00681-18
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