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Taxol Analogues Exhibit Differential Effects on Photoaffinity Labeling of β-Tubulin and the Multidrug Resistance Associated P-Glycoprotein

Several next-generation taxanes have been reported to possess high potency against Taxol-resistant cancer cell lines overexpressing βIII-tubulin and/or P-glycoprotein (P-gp), both of which are involved in drug resistance. Using a photoaffinity Taxol analogue, 2-(m-azidobenzoyl)-taxol, two potent nex...

पूर्ण विवरण

में बचाया:
ग्रंथसूची विवरण
में प्रकाशित:J Nat Prod
मुख्य लेखकों: Yang, Chia-Ping Huang, Wang, Changwei, Ojima, Iwao, Horwitz, Susan Band
स्वरूप: Artigo
भाषा:Inglês
प्रकाशित: 2018
विषय:
ऑनलाइन पहुंच:https://ncbi.nlm.nih.gov/pmc/articles/PMC6147140/
https://ncbi.nlm.nih.gov/pubmed/29517223
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jnatprod.7b01047
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