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Designing novel inhibitors against Mycobacterium tuberculosis FadA5 (acetyl-CoA acetyltransferase) by virtual screening of known anti-tuberculosis (bioactive) compounds

By-products of fatty acid degradation are extensively utilized by Mycobacterium tuberculosis (Mtb) for lipid synthesis and energy production during the infection phase. Cholesterol from host is scavenged by Mtb to fulfill its metabolic requirements, evade host immunity and invade macrophages. Blocki...

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Publicat a:Bioinformation
Autors principals: Jaiswal, Atul Kumar, Husaini, Syed Hussain Abbas, Kumar, Amarjeet, Subbarao, Naidu
Format: Artigo
Idioma:Inglês
Publicat: Biomedical Informatics 2018
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6137569/
https://ncbi.nlm.nih.gov/pubmed/30237678
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.6026/97320630014327
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