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Drug permeation and metabolism in Mycobacterium tuberculosis: prioritising local exposure as essential criterion in new TB drug development

Anti-tuberculosis (TB) drugs possess diverse abilities to penetrate the different host tissues and cell types in which infecting Mycobacterium tuberculosis bacilli are located during active disease. This is important since there is increasing evidence that the respective “lesion-penetrating” propert...

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Detalles Bibliográficos
Publicado en:IUBMB Life
Main Authors: Tanner, Lloyd, Denti, Paolo, Wiesner, Lubbe, Warner, Digby F.
Formato: Artigo
Idioma:Inglês
Publicado: 2018
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC6129860/
https://ncbi.nlm.nih.gov/pubmed/29934964
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/iub.1866
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