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Structural Plasticity in the C‑Terminal Region of Macrophage Migration Inhibitory Factor‑2 Is Associated with an Induced Fit Mechanism for a Selective Inhibitor

We report the first reversible and selective small molecule inhibitor of pro-inflammatory protein macrophage migration inhibitory factor-2 (also known as MIF-2 or D-DT). 4-(3-Carboxyphenyl)-2,5pyridinedicarboxylic acid (4-CPPC) shows competitive binding with a 13fold selectivity for human MIF-2 vers...

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Detalhes bibliográficos
Publicado no:Biochemistry
Main Authors: Pantouris, Georgios, Bucala, Richard, Lolis, Elias J.
Formato: Artigo
Idioma:Inglês
Publicado em: 2018
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6123015/
https://ncbi.nlm.nih.gov/pubmed/29847104
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.biochem.8b00344
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