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Cooperative recognition of T:T mismatch by echinomycin causes structural distortions in DNA duplex

Small-molecule compounds that target mismatched base pairs in DNA offer a novel prospective for cancer diagnosis and therapy. The potent anticancer antibiotic echinomycin functions by intercalating into DNA at CpG sites. Surprisingly, we found that the drug strongly prefers to bind to consecutive Cp...

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Dettagli Bibliografici
Pubblicato in:Nucleic Acids Res
Autori principali: Wu, Pei-Ching, Tzeng, Shu-Ling, Chang, Chung-ke, Kao, Ya-Fen, Waring, Michael J, Hou, Ming-Hon
Natura: Artigo
Lingua:Inglês
Pubblicazione: Oxford University Press 2018
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6101601/
https://ncbi.nlm.nih.gov/pubmed/29741655
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1093/nar/gky345
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