Yüklüyor......

Synthesis and PI3 Kinase Inhibition Activity of a Wortmannin-Leucine Derivative

Wortmannin is a potent covalent inhibitor of PI3K that shows substantial in vivo toxicity and thus is unsuitable for systemic therapeutic applications. One possible approach to minimize systemic toxicity is to generate a latent wortmannin pro-drug that will be selectively activated in target tissues...

Ful tanımlama

Kaydedildi:
Detaylı Bibliyografya
Yayımlandı:Molecules
Asıl Yazarlar: Cantrell, William, Huang, Yue, Menchaca, Antonio A., Kulik, George, Welker, Mark E.
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: MDPI 2018
Konular:
Online Erişim:https://ncbi.nlm.nih.gov/pmc/articles/PMC6100554/
https://ncbi.nlm.nih.gov/pubmed/30036994
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules23071791
Etiketler: Etiketle
Etiket eklenmemiş, İlk siz ekleyin!