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Analogue Synthesis Reveals Decoupling of Antibiofilm and β-Lactam Potentiation Activities of a Lead 2-Aminoimidazole Adjuvant Against Mycobacterium smegmatis

Biofilm formation is one of the many mechanisms bacteria utilize to survive antibiotic treatment. It has been demonstrated that when Mycobacterium tuberculosis exists in a biofilm in vitro it expresses phenotypic resistance to antimicrobial drugs. Since the in vivo survival of M. tuberculosis follow...

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Publicat a:Chem Biol Drug Des
Autors principals: Martin, Sara E., Nguyen, Catherine M., Basaraba, Randall J., Melander, Christian
Format: Artigo
Idioma:Inglês
Publicat: 2018
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6097888/
https://ncbi.nlm.nih.gov/pubmed/29663670
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/cbdd.13208
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