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Quantitative and Mechanistic Understanding of AZD1775 Penetration across Human Blood–Brain Barrier in Glioblastoma Patients Using an IVIVE–PBPK Modeling Approach

PURPOSE: AZD1775, a first-in-class, small-molecule inhibitor of the Wee1 tyrosine kinase, is under evaluation as a potential chemo- and radiosensitizer for treating glioblastoma. This study was to prospectively, quantitatively, and mechanistically investigate the penetration of AZD1775 across the hu...

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Publicat a:Clin Cancer Res
Autors principals: Li, Jing, Wu, Jianmei, Bao, Xun, Honea, Norissa, Xie, Youming, Kim, Seongho, Sparreboom, Alex, Sanai, Nader
Format: Artigo
Idioma:Inglês
Publicat: 2017
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6097184/
https://ncbi.nlm.nih.gov/pubmed/28928160
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1158/1078-0432.CCR-17-0983
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