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Orthoester functionalized N-guanidino derivatives of 1,5-dideoxy-1,5-imino-d-xylitol as pH-responsive inhibitors of β-glucocerebrosidase

Alkylated guanidino derivatives of 1,5-dideoxy-1,5-imino-d-xylitol bearing an orthoester moiety were prepared using a concise synthetic protocol. Inhibition assays with a panel of glycosidases revealed that one of the compounds prepared displays potent inhibition against human β-glucocerebrosidase (...

Ausführliche Beschreibung

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Bibliographische Detailangaben
Veröffentlicht in:Medchemcomm
Hauptverfasser: Sevšek, Alen, Sastre Toraño, Javier, Quarles van Ufford, Linda, Moret, Ed E., Pieters, Roland J., Martin, Nathaniel I.
Format: Artigo
Sprache:Inglês
Veröffentlicht: Royal Society of Chemistry 2017
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC6072142/
https://ncbi.nlm.nih.gov/pubmed/30108721
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c7md00480j
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