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Farnesyltransferase-mediated Delivery of a Covalent Inhibitor Overcomes Alternative Prenylation to Mislocalize K-Ras

Mutationally activated Ras is one of the most common oncogenic drivers found across all malignancies, and its selective inhibition has long been a goal in both pharma and academia. One of the oldest and most validated methods to inhibit overactive Ras signaling is by interfering with its post-transl...

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Pubblicato in:ACS Chem Biol
Autori principali: Novotny, Chris J., Hamilton, Gregory L., McCormick, Frank, Shokat, Kevan M.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2017
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6070134/
https://ncbi.nlm.nih.gov/pubmed/28530791
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acschembio.7b00374
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