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Sodium Diisopropylamide in Tetrahydrofuran: Selectivities, Rates, and Mechanisms of Arene Metalations

Sodium diisopropylamide (NaDA)-mediated metalations of arenes in tetrahydrofuran (THF)/hexane or THF/Me(2)NEt solutions are described. A survey of >40 benzenoid- and pyridine-based arenes with a range of substituents demonstrates the efficacy and regioselectivity of metalation. Metalations of act...

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Bibliografiset tiedot
Julkaisussa:J Am Chem Soc
Päätekijät: Algera, Russell F., Ma, Yun, Collum, David B.
Aineistotyyppi: Artigo
Kieli:Inglês
Julkaistu: 2017
Aiheet:
Linkit:https://ncbi.nlm.nih.gov/pmc/articles/PMC6059610/
https://ncbi.nlm.nih.gov/pubmed/28946744
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jacs.7b08734
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