A carregar...

Glutamic acid–valine–citrulline linkers ensure stability and efficacy of antibody–drug conjugates in mice

Valine–citrulline linkers are commonly used as enzymatically cleavable linkers for antibody–drug conjugates. While stable in human plasma, these linkers are unstable in mouse plasma due to susceptibility to an extracellular carboxylesterase. This instability often triggers premature release of drugs...

ver descrição completa

Na minha lista:
Detalhes bibliográficos
Publicado no:Nat Commun
Main Authors: Anami, Yasuaki, Yamazaki, Chisato M., Xiong, Wei, Gui, Xun, Zhang, Ningyan, An, Zhiqiang, Tsuchikama, Kyoji
Formato: Artigo
Idioma:Inglês
Publicado em: Nature Publishing Group UK 2018
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6023893/
https://ncbi.nlm.nih.gov/pubmed/29955061
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41467-018-04982-3
Tags: Adicionar Tag
Sem tags, seja o primeiro a adicionar uma tag!