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Investigation of piperazines as human carbonic anhydrase I, II, IV and VII activators

Four human (h) carbonic anhydrase isoforms (CA, EC 4.2.1.1), hCA I, II, IV, and VII, were investigated for their activation profile with piperazines belonging to various classes, such as N-aryl-, N-alkyl-, N-acyl-piperazines as well as 2,4-disubstituted derivatives. As the activation mechanism invol...

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Dettagli Bibliografici
Pubblicato in:J Enzyme Inhib Med Chem
Autori principali: Angeli, Andrea, Chiaramonte, Niccolò, Manetti, Dina, Romanelli, Maria Novella, Supuran, Claudiu T.
Natura: Artigo
Lingua:Inglês
Pubblicazione: Taylor & Francis 2017
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6009915/
https://ncbi.nlm.nih.gov/pubmed/29280407
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1080/14756366.2017.1417277
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