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Extending in Silico Protein Target Prediction Models to Include Functional Effects

In silico protein target deconvolution is frequently used for mechanism-of-action investigations; however existing protocols usually do not predict compound functional effects, such as activation or inhibition, upon binding to their protein counterparts. This study is hence concerned with including...

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Dades bibliogràfiques
Publicat a:Front Pharmacol
Autors principals: Mervin, Lewis H., Afzal, Avid M., Brive, Lars, Engkvist, Ola, Bender, Andreas
Format: Artigo
Idioma:Inglês
Publicat: Frontiers Media S.A. 2018
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6004408/
https://ncbi.nlm.nih.gov/pubmed/29942259
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3389/fphar.2018.00613
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