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A “Cross-Stitched” Peptide with Improved Helicity and Proteolytic Stability

A new computational approach to obtain quantitative energy profiles for helix folding was used in the design of orthogonal hydrocarbon and lactam bicyclic peptides. The proteolytically stable,“cross-stitched” peptide SRC2-BCP1 shows nanomolar affinity for estrogen receptor α and x-ray crystallograph...

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Detalles Bibliográficos
Publicado en:Org Biomol Chem
Main Authors: Speltz, Thomas E., Mayne, Christopher G., Fanning, Sean W., Siddiqui, Zamia, Tajkhorshid, Emad, Greene, Geoffrey L., Moore, Terry W.
Formato: Artigo
Idioma:Inglês
Publicado: 2018
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC5993042/
https://ncbi.nlm.nih.gov/pubmed/29725689
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c8ob00790j
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