A “Cross-Stitched” Peptide with Improved Helicity and Proteolytic Stability

Por Speltz, Thomas E., Mayne, Christopher G., Fanning, Sean W., Siddiqui, Zamia, Tajkhorshid, Emad, Greene, Geoffrey L., Moore, Terry W.
Publicado no Org Biomol Chem (2018)

Replacement of a Naphthalene Scaffold in Kelch-like ECH-Associated Protein 1 (KEAP1)/ Nuclear factor (erythroid-derived 2)-like 2 (NRF2) Inhibitors

Por Richardson, Benjamin G., Jain, Atul D., Potteti, Haranatha, Lazzara, Phillip R., David, Brian P., Tamatam, Chandra, Choma, Ewelina, Skowron, Kornelia, Dye, Katherine, Siddiqui, Zamia, Wang, Yue-Ting, Krunic, Aleksej, Reddy, Sekhar P., Moore, Terry W.
Publicado no J Med Chem (2018)