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An efficient new method for the synthesis of 3-[(18)F]fluoro-4-aminopyridine via Yamada-Curtius rearrangement
4-Aminopyridine is a clinically approved drug to improve motor symptoms in multiple sclerosis. A fluorine-18-labeled derivative of this drug, 3-[(18)F]fluoro-4-aminopyridine, is currently under investigation for positron emission tomography (PET) imaging of demyelination. Herein, the Yamada-Curtius...
Kaydedildi:
Yayımlandı: | J Labelled Comp Radiopharm |
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Asıl Yazarlar: | , , , , |
Materyal Türü: | Artigo |
Dil: | Inglês |
Baskı/Yayın Bilgisi: |
2017
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Konular: | |
Online Erişim: | https://ncbi.nlm.nih.gov/pmc/articles/PMC5992582/ https://ncbi.nlm.nih.gov/pubmed/28870001 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/jlcr.3560 |
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