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α‐Conotoxins active at α3‐containing nicotinic acetylcholine receptors and their molecular determinants for selective inhibition

Neuronal α3‐containing nicotinic acetylcholine receptors (nAChRs) in the peripheral nervous system (PNS) and non‐neuronal tissues are implicated in a number of severe disease conditions ranging from cancer to cardiovascular diseases and chronic pain. However, despite the physiological characterizati...

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Détails bibliographiques
Publié dans:Br J Pharmacol
Auteurs principaux: Cuny, Hartmut, Yu, Rilei, Tae, Han‐Shen, Kompella, Shiva N, Adams, David J
Format: Artigo
Langue:Inglês
Publié: John Wiley and Sons Inc. 2017
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC5979624/
https://ncbi.nlm.nih.gov/pubmed/28477355
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/bph.13852
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