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Artificial macrocycles as IL-17A/IL-17RA antagonists

Interleukin 17(A) is a pro-inflammatory cytokine involved in several auto-immune and inflammatory diseases. Current antagonists against IL-17(A) or its receptor (IL-17RA) that show efficacy in clinical trials are monoclonal antibodies (mAbs). However, recently designed artificial macrocycles are pot...

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Detalhes bibliográficos
Publicado no:Medchemcomm
Main Authors: Wang, Wenjia, Groves, Matthew R., Dömling, Alexander
Formato: Artigo
Idioma:Inglês
Publicado em: Royal Society of Chemistry 2017
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5937545/
https://ncbi.nlm.nih.gov/pubmed/29750108
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c7md00464h
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