Carregant...

Antitumor Activity of a Novel Quinoline Derivative, TAS‐103, with Inhibitory Effects on Topoisomerases I and II

A novel quinoline derivative, TAS‐103 (6‐[[2‐(dimethyIamino)ethyl]amino]‐3‐hydroxy‐7H‐indeno[2,l‐c]quinolin‐7‐one dihydrochloride), was developed as an anticancer agent targeting topoisomerases (topo) I and II, with marked efficacy in solid tumors. TAS‐103 inhibited topo I and II (IC(50): 2 μM, 6.5...

Descripció completa

Guardat en:
Dades bibliogràfiques
Publicat a:Jpn J Cancer Res
Autors principals: Utsugi, Teruhiro, Aoyagi, Kumio, Asao, Tetsuji, Okazaki, Shinji, Aoyagi, Yoshimi, Sano, Masaki, Wierzba, Konstanty, Yamada, Yuji
Format: Artigo
Idioma:Inglês
Publicat: Blackwell Publishing Ltd 1997
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC5921285/
https://ncbi.nlm.nih.gov/pubmed/9414662
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/j.1349-7006.1997.tb00320.x
Etiquetes: Afegir etiqueta
Sense etiquetes, Sigues el primer a etiquetar aquest registre!