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Sialidase-catalyzed one-pot multienzyme (OPME) synthesis of sialidase transition-state analogue inhibitors

Sialidase transition state analog inhibitor 2,3-dehydro-2-deoxy-N-acetylneuraminic acid (Neu5Ac2en, DANA) has played a leading role in developing clinically used anti-influenza virus drugs. Taking advantage of the Neu5Ac2en-forming catalytic property of Streptococcus pneumoniae sialidase SpNanC, an...

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Detalhes bibliográficos
Publicado no:ACS Catal
Main Authors: Xiao, An, Li, Yanhong, Li, Xixuan, Santra, Abhishek, Yu, Hai, Li, Wanqing, Chen, Xi
Formato: Artigo
Idioma:Inglês
Publicado em: 2017
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5920526/
https://ncbi.nlm.nih.gov/pubmed/29713561
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acscatal.7b03257
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