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Pharmacokinetics and interspecies scaling of a novel, orally-bioavailable anti-cancer drug, SHetA2

SHetA2 is a small molecule drug with promising cancer prevention and therapeutic activity and a high preclinical safety profile. The study objectives were to perform interspecies scaling and pharmacokinetic (PK) modeling of SHetA2 for human PK prediction. The PK data obtained from mice, rats, and do...

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Pubblicato in:PLoS One
Autori principali: Sharma, Ankur, Benbrook, Doris Mangiaracina, Woo, Sukyung
Natura: Artigo
Lingua:Inglês
Pubblicazione: Public Library of Science 2018
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5892888/
https://ncbi.nlm.nih.gov/pubmed/29634717
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1371/journal.pone.0194046
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