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The plant sesquiterpene lactone parthenolide inhibits Wnt/β-catenin signaling by blocking synthesis of the transcriptional regulators TCF4/LEF1

The Wnt/β-catenin pathway is essential for embryonic development and homeostasis, but excessive activation of this pathway is frequently observed in various human diseases, including cancer. Current therapeutic drugs targeting the Wnt pathway often lack sufficient efficacy, and new compounds targeti...

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Publicado en:J Biol Chem
Autores principales: Zhu, Xiaoliang, Yuan, Chunmao, Tian, Chenyang, Li, Chen, Nie, Fen, Song, Xiaomin, Zeng, Rong, Wu, Dianqing, Hao, Xiaojiang, Li, Lin
Formato: Artigo
Lenguaje:Inglês
Publicado: American Society for Biochemistry and Molecular Biology 2018
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC5892590/
https://ncbi.nlm.nih.gov/pubmed/29462785
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1074/jbc.M117.819300
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