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Modeling and resistant alleles explain the selectivity of antimalarial compound 49c towards apicomplexan aspartyl proteases

Toxoplasma gondii aspartyl protease 3 (TgASP3) phylogenetically clusters with Plasmodium falciparum Plasmepsins IX and X (PfPMIX, PfPMX). These proteases are essential for parasite survival, acting as key maturases for secreted proteins implicated in invasion and egress. A potent antimalarial peptid...

Täydet tiedot

Tallennettuna:
Bibliografiset tiedot
Julkaisussa:EMBO J
Päätekijät: Mukherjee, Budhaditya, Tessaro, Francesca, Vahokoski, Juha, Kursula, Inari, Marq, Jean‐Baptiste, Scapozza, Leonardo, Soldati‐Favre, Dominique
Aineistotyyppi: Artigo
Kieli:Inglês
Julkaistu: John Wiley and Sons Inc. 2018
Aiheet:
Linkit:https://ncbi.nlm.nih.gov/pmc/articles/PMC5881632/
https://ncbi.nlm.nih.gov/pubmed/29519896
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.15252/embj.201798047
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