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Dynamic rearrangement of the intrinsic ligand regulates KCNH potassium channels

KCNH voltage-gated potassium channels (EAG, ERG, and ELK) play significant roles in neuronal and cardiac excitability. They contain cyclic nucleotide-binding homology domains (CNBHDs) but are not directly regulated by cyclic nucleotides. Instead, the CNBHD ligand-binding cavity is occupied by an int...

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Detalhes bibliográficos
Publicado no:J Gen Physiol
Main Authors: Dai, Gucan, James, Zachary M., Zagotta, William N.
Formato: Artigo
Idioma:Inglês
Publicado em: Rockefeller University Press 2018
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5881448/
https://ncbi.nlm.nih.gov/pubmed/29567795
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1085/jgp.201711989
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