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An Inexpensive, In-House-Made, Microdialysis Device for Measuring Drug–Protein Binding

[Image: see text] An inexpensive, in-house made microdialysis device is described that is suitable for measuring the binding of small molecules including drug candidates to serum proteins or other macromolecules. The device is based on the standard equilibrium dialysis method to measure the fraction...

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Pubblicato in:ACS Med Chem Lett
Autori principali: Herbst, Zackary M., Shibata, Sayaka, Fan, Erkang, Gelb, Michael H.
Natura: Artigo
Lingua:Inglês
Pubblicazione: American Chemical Society 2017
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5846030/
https://ncbi.nlm.nih.gov/pubmed/29541374
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsmedchemlett.7b00316
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