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Study of Interactions of an Anticancer Drug Neratinib With Bovine Serum Albumin: Spectroscopic and Molecular Docking Approach

Binding of therapeutic agents to plasma proteins, particularly to serum albumin, provides valuable information in the drug development. This study was designed to evaluate the binding interaction of neratinib with bovine serum albumin (BSA). Neratinib blocks HER2 signaling and is effective in trastu...

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Pubblicato in:Front Chem
Autori principali: Wani, Tanveer A., Bakheit, Ahmed H., Abounassif, M. A., Zargar, Seema
Natura: Artigo
Lingua:Inglês
Pubblicazione: Frontiers Media S.A. 2018
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5845959/
https://ncbi.nlm.nih.gov/pubmed/29564326
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3389/fchem.2018.00047
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