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Integrated In Silico Fragment-Based Drug Design: Case Study with Allosteric Modulators on Metabotropic Glutamate Receptor 5

GPCR allosteric modulators target at the allosteric binding pockets of G protein-coupled receptors (GPCRs) with indirect influence on the effects of an orthosteric ligand. Such modulators exhibit significant advantages compared to the corresponding orthosteric ligands, including better chemical trac...

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Detalles Bibliográficos
Publicado en:AAPS J
Main Authors: Bian, Yuemin, Feng, Zhiwei, Yang, Peng, Xie, Xiang-Qun
Formato: Artigo
Idioma:Inglês
Publicado: 2017
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC5836546/
https://ncbi.nlm.nih.gov/pubmed/28560482
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1208/s12248-017-0093-5
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