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Synthesis of N-alkoxy-substituted 2H-benzimidazoles

Treatment of 2-nitro-N-(2-methyl-1-propen-1-yl)benzenamines with potassium tert-butoxide in tert-butanol followed by the addition of an electrophile affords N-alkoxy-2H-benzimidazoles. Electrophiles including methyl iodide, allylic bromides, propargylic bromides, benzyl bromide, and acetyl chloride...

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Detalles Bibliográficos
Publicado en:Tetrahedron Lett
Autores principales: Ansari, Nurul H., Söderberg, Björn C. G.
Formato: Artigo
Lenguaje:Inglês
Publicado: 2017
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC5830180/
https://ncbi.nlm.nih.gov/pubmed/29503480
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.tetlet.2017.11.007
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