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Improving Therapeutic Potential of Farnesylthiosalicylic Acid: Tumor Specific Delivery via Conjugation with Heptamethine Cyanine Dye

The RAS and mTOR inhibitor S-trans-trans-farnesylthiosalicylic acid (FTS) is a promising anticancer agent with moderate potency, currently undergoing clinical trials as a chemotherapeutic agent. FTS has displayed its potential against a variety of cancers including endocrine resistant breast cancer....

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Publicat a:Mol Pharm
Autors principals: Guan, Yang, Zhang, Yi, Xiao, Li, Li, Jie, Wang, Ji-ping, Chordia, Mahendra D., Liu, Zhong-Qiu, Chung, Leland W. K., Yue, Wei, Pan, Dongfeng
Format: Artigo
Idioma:Inglês
Publicat: 2016
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC5815365/
https://ncbi.nlm.nih.gov/pubmed/26992462
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.molpharmaceut.5b00906
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