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Antibacterial Evaluation and Virtual Screening of New Thiazolyl-Triazole Schiff Bases as Potential DNA-Gyrase Inhibitors

The global spread of bacterial resistance to drugs used in therapy requires new potent and safe antimicrobial agents. DNA gyrases represent important targets in drug discovery. Schiff bases, thiazole, and triazole derivatives are considered key scaffolds in medicinal chemistry. Fifteen thiazolyl-tri...

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Detaylı Bibliyografya
Yayımlandı:Int J Mol Sci
Asıl Yazarlar: Nastasă, Cristina, Vodnar, Dan C., Ionuţ, Ioana, Stana, Anca, Benedec, Daniela, Tamaian, Radu, Oniga, Ovidiu, Tiperciuc, Brînduşa
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: MDPI 2018
Konular:
Online Erişim:https://ncbi.nlm.nih.gov/pmc/articles/PMC5796171/
https://ncbi.nlm.nih.gov/pubmed/29324679
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ijms19010222
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