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Antibacterial Evaluation and Virtual Screening of New Thiazolyl-Triazole Schiff Bases as Potential DNA-Gyrase Inhibitors

The global spread of bacterial resistance to drugs used in therapy requires new potent and safe antimicrobial agents. DNA gyrases represent important targets in drug discovery. Schiff bases, thiazole, and triazole derivatives are considered key scaffolds in medicinal chemistry. Fifteen thiazolyl-tri...

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Detalhes bibliográficos
Publicado no:Int J Mol Sci
Main Authors: Nastasă, Cristina, Vodnar, Dan C., Ionuţ, Ioana, Stana, Anca, Benedec, Daniela, Tamaian, Radu, Oniga, Ovidiu, Tiperciuc, Brînduşa
Formato: Artigo
Idioma:Inglês
Publicado em: MDPI 2018
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5796171/
https://ncbi.nlm.nih.gov/pubmed/29324679
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ijms19010222
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