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Peptidomimetic therapeutics: scientific approaches and opportunities

Natural endogenously occurring peptides exhibit desirable medicinal properties, but are often limited in application by rapid proteolysis and inadequate membrane permeability. However, editing naturally occurring peptide sequences to develop peptidomimetic analogs created a promising class of therap...

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Detalhes bibliográficos
Publicado no:Drug Discov Today
Main Authors: Qvit, Nir, Rubin, Samuel J.S., Urban, Travis J., Mochly-Rosen, Daria, Gross, Eric R.
Formato: Artigo
Idioma:Inglês
Publicado em: 2016
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5759319/
https://ncbi.nlm.nih.gov/pubmed/27856346
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.drudis.2016.11.003
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