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Molecular Docking and 3D-Pharmacophore Modeling to Study the Interactions of Chalcone Derivatives with Estrogen Receptor Alpha

Tamoxifen is the most frequently used anti-estrogen adjuvant treatment for estrogen receptor-positive breast cancer. However, it is associated with an increased risk of several serious side–effects, such as uterine cancer, stroke, and pulmonary embolism. The 2′,4′-dihydroxy-6-methoxy-3,5-dimethylcha...

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Detalhes bibliográficos
Publicado no:Pharmaceuticals (Basel)
Main Authors: Muchtaridi, Muchtaridi, Syahidah, Hasna Nur, Subarnas, Anas, Yusuf, Muhammad, Bryant, Sharon D., Langer, Thierry
Formato: Artigo
Idioma:Inglês
Publicado em: MDPI 2017
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5748638/
https://ncbi.nlm.nih.gov/pubmed/29035298
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ph10040081
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