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Identification and characterization of the structure–activity relationships involved in UGT1A1 inhibition by anthraquinone and dianthrone constituents of Polygonum multiflorum

The adverse effects of Polygonum (P.) multiflorum, including abnormal bilirubin metabolism, are a serious public health issue. As uridine diphosphate (UDP)-glucuronosyltransferase 1A1 (UGT1A1) is the only enzyme responsible for bilirubin metabolism, we investigated the inhibitory effect of a P. mult...

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Enregistré dans:
Détails bibliographiques
Publié dans:Sci Rep
Auteurs principaux: Wang, Qi, Wang, Yadan, Li, Yong, Wen, Binyu, Dai, Zhong, Ma, Shuangcheng, Zhang, Yujie
Format: Artigo
Langue:Inglês
Publié: Nature Publishing Group UK 2017
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC5738440/
https://ncbi.nlm.nih.gov/pubmed/29263357
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41598-017-18231-y
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